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6-tetra-O-acteyl-1-C-[4-chloro-3-[[4-[[(3S)-tetrahydrofu-ran-3-yl]oxy]phenyl]

6-tetra-O-acteyl-1-C-[4-chloro-3-[[4-[[(3S)-tetrahydrofu-ran-3-yl]oxy]phenyl]

Incazelo emfushane:

Ifomula yemolekyuli:C31H35ClO11
Isisindo se-molecule: 619.056
Inombolo ye-CAS:915095-99-7


Imininingwane Yomkhiqizo

Omaka bomkhiqizo

Isicelo

Lo mkhiqizo uyithebhulethi ekhanyayo ephuzi ehlanganiswe nefilimu, emhlophe noma ecishe ibe mhlophe ngemva kokukhipha okunamathelayo.

Izinkomba
Lo mkhiqizo ulungele ukwelapha isifo sikashukela sohlobo 2.

I-Monotherapy
Lo mkhiqizo usetshenziswa ngokuhambisana nokulawulwa kokudla kanye nokuzivocavoca ukuze kuthuthukiswe ukulawula ushukela wegazi ezigulini ezinesifo sikashukela sohlobo 2.

Isetshenziswa ngokuhlanganiswa ne-metformin hydrochloride
Lapho i-metformin hydrochloride iyodwa ingakwazi ukulawula ushukela wegazi ngempumelelo, lo mkhiqizo ungasetshenziswa uhlanganiswe ne-metformin hydrochloride ukuthuthukisa ukulawulwa kokushukela ezigulini ezinesifo sikashukela sohlobo 2 ngesisekelo sokudla nokuzivocavoca umzimba.

Isetshenziswa ngokuhlanganiswa ne-metformin hydrochloride kanye ne-sulfonylureas.
Lapho ukusetshenziswa okuhlangene kwe-metformin hydrochloride kanye ne-sulfonylureas kungakwazi ukulawula ushukela wegazi ngempumelelo, lo mkhiqizo ungasetshenziswa uhlanganiswe ne-metformin hydrochloride kanye ne-sulfonylureas ukuthuthukisa ukulawula ushukela wegazi ezigulini ezinesifo sikashukela sohlobo 2 ngesisekelo sokudla nokuzivocavoca.

Imikhawulo yemithi
Lo mkhiqizo awunconywa ezigulini ezinesifo sikashukela sohlobo loku-1 noma ekwelapheni i-ketoacidosis yesifo sikashukela.

Ukucaciswa
(1) 10 mg;(2) 25 mg.

Umthamo
Umthamo onconyiwe.
Umthamo onconyiwe walo mkhiqizo ngu-10 mg ekuseni, kanye ngosuku, esiswini esingenalutho noma ngemva kokudla.Ezigulini ezibekezelela lo mkhiqizo, umthamo unganyuswa ube ngu-25 mg (bona [Izilingo Zomtholampilo]).
Ezigulini ezine-hypovolemia, kunconywa ukuthi kulungiswe i-hypovolemia ngaphambi kokuqala ukusebenzisa lo mkhiqizo (bona [Izixwayiso]).

Iziguli ezinokukhubazeka kwezinso.
Kunconywa ukuhlola ukusebenza kwezinso ngaphambi kokuqala ukusebenzisa lo mkhiqizo, bese kufanele uhlolwe njalo.
Iziguli i-eGFR yazo ingaphansi kuka-45 mL/min/1.73 m2 akufanele zisebenzise lo mkhiqizo.
Iziguli ezine-eGFR ephakeme noma elingana no-45 mL/min/1.73 m2 azidingi ukulungisa umthamo.
Uma i-eGFR ilokhu ingaphansi kuka-45 mL/min/1.73 m2, lo mkhiqizo kufanele uyekwe (bona [Izixwayiso]).

Iziguli ezinokulimala kwesibindi.
Iziguli ezinokulimala kwesibindi azidingi ukulungisa umthamo.Ukuchayeka kwe-Enpagliflozin kukhuphuke ezigulini ezinokulimala okukhulu kwesibindi.Isipiliyoni sokwelashwa kweziguli ezinokulimala okukhulu kwesibindi sinqunyelwe, ngakho-ke, akunconywa kule ngxenye yabantu.

Okujwayelekile:izinga lebhizinisi
ubumsulwa:≥99.0%

Ingaphandle:impushana emhlophe ukuya emhlophe
Iphakheji:25kg/isigubhu

Ulayini Womkhiqizo Ohlanganisiwe Wezinsiza

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Isitifiketi

I-JIN DUN Medical ineIziqu ze-ISO futhi ihlangabezana namazinga okukhiqiza e-GMP, kuqashwe ochwepheshe basekhaya nabangaphandle abanolwazi olunzulu lokuqondisa i-R&D yenkampani.

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Izinzuzo Zokwenza Ngokwezifiso Kwezokwelapha

TECHNOL OGY UBUHLE
●I-High Pressure Catalytic Hydrogenation.I-High Pressure Hydrogenolysis Reaction .Ukusabela kwe-Cryogenic (<-78%C)
● I-Aromatic Heterocyclic Synthesis
●Ukusabela Kabusha
●Chiral Resolution
●Heck, Suzuki,Negishi,Sonogashira .Ukusabela kukaGiignard

I-JIN DUN R&D

Izisetshenziswa

Ilebhu yethu inezinsiza ezihlukahlukene zokuhlola nokuhlola, njenge: NMR (Bruker 400M), HPLC、chiral-HPLC、LC-MS、LC-MS/MS (API 4000),IR,UV,GC,GC,GC-MS, Chromatography, I-Microwave Synthesizer, i-Parallel Synthesizer, i-Differential Scanning Calorimeter (DSC), i-Electron Microscope...

Ithimba le-R&D

I-Jindun Medical ineqembu labasebenzi abangochwepheshe be-R&D, futhi isebenzisa ochwepheshe abaningi bokwenziwa kwezidakamizwa basekhaya nabangaphandle ukuze baqondise i-R&D, okwenza ukuhlanganiswa kwethu kunembe kakhudlwana futhi kusebenze kahle.

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Ukwabelana Kwamacala

Sisize izinkampani ezimbalwa eziphezulu zasekhaya ezithaka imithi, njengeI-Hansoh, i-Hengrui ne-HEC Pharm.Lapha sizokhombisa ingxenye yazo.

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Ikesi Lokwenza Ngokwezifiso:

Inombolo yeCas: 110351-94-5

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Ikesi Lokwenza Ngokwezifiso:

Inombolo yeCas: 144848-24-8

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Ikesi Lesithathu Lokwenza Ngokwezifiso:

Inombolo yeCas: 200636-54-0

Imodi Yokubambisana

1.Enza ngendlela oyifisayo i-New Intermediates noma ama-API.Ngokufanayo nokwabelana kwecala elingenhla, amakhasimende anezidingo ze-Intermediates ethile noma ama-API, futhi awakwazi ukuthola imikhiqizo edingekayo emakethe, lapho-ke singasiza Ukwenza Ngokwezifiso.

2.Ukuthuthukisa Inqubo Yemikhiqizo Emidala.Ithimba lethu lizosiza Ukuthuthukisa futhi lithuthukise ukukhiqiza okunjalo okuyindlela yokusabela endala, izindleko zokukhiqiza ziphezulu, nokusebenza kahle kuphansi.Singahlinzeka ngemibhalo egcwele yokudluliswa kobuchwepheshe kanye nokuthuthukiswa kwenqubo, sisize ikhasimende ngokukhiqiza okuphumelelayo.

Ukusuka kokuhlosiwe kwezidakamizwa kuye kuma-IND, i-JIN DUN Medical ikunikezaizixazululo zomuntu siqu ze-R&D zokuma okukodwa.

I-JIN DUN Medical iphikelela ekwakheni iqembu elinamaphupho, ukwenza imikhiqizo enesizotha, ecophelelayo, eqinile, futhi siphume konke ukuze sibe uzakwethu othembekile nomngane wamakhasimende!


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