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I-OEM Customized Rivaroxaban CAS No.

I-OEM Customized Rivaroxaban CAS No.

Incazelo emfushane:

Ifomula yemolekyuli: C19H18ClN3O5S

Isisindo samangqamuzana: 435.88

I-CAS no: 366789-02-8


Imininingwane Yomkhiqizo

Omaka bomkhiqizo

Imikhiqizo yethu ibhekwa kabanzi futhi ithembekile kubasebenzisi bokugcina futhi ingahlangabezana nezidingo ezihlala zishintsha zezimali nezenhlalo ze-OEM Customized Rivaroxaban CAS No. ukuthambekela kokuthuthukiswa kwale mboni futhi ugcwalise injabulo yakho ngempumelelo.Kunoma ubani othathekayo ngaphakathi kwezixazululo zethu, kufanele uxhumane nathi ngokukhululekile.
Imikhiqizo yethu ibhekwa kabanzi futhi ithembekile kubasebenzisi bokugcina futhi ingahlangabezana nezidingo ezihlala zishintsha zezimali nezenhlaloI-China Chemical and Pharmaceutical Raw Material, Sinezixazululo ezingcono kakhulu kanye nokuthengisa okufanelekayo kanye nethimba lobuchwepheshe.Ngokuthuthukiswa kwenkampani yethu, siyakwazi ukuletha amakhasimende imikhiqizo engcono kakhulu, ukusekelwa okuhle kwezobuchwepheshe, isevisi ephelele emva kokuthengisa.

Isetshenziswa ezigulini ezikhulile ezinokuhlinzwa okukhethiwe kwe-hip noma idolo ukuvimbela i-venous thrombosis (VTE).

Isetshenziselwa ukuvimbela noma ukunciphisa ukwakheka kwe-thrombosis, i-deep vein thrombosis (DVT) kanye ne-pulmonary embolism (PE) ngemva kokuhlinzwa esikhundleni se-hip noma amadolo.

Umthamo onconyiwe yi-rivaroxaban yomlomo 10mg, kanye ngosuku.I-Rivaroxaban 10mg ingathathwa ngokudla noma yodwa.I-Rivaroxaban 15mg noma amaphilisi angu-20mg kufanele athathwe nokudla.

standard: usp40
Isilinganiso: 99-102%

Ingaphandle: Impushana emhlophe
Iphakheji: 25kg / isigubhu

Thatha 4-(4-aminophenyl) morpholin-3-one (SM-1), (S)-N-glycidyl phthalimide (SM-2), 5-chlorothiophene-2- Formyl chloride (SM-3) into yokuqala .Ngemuva kwe-condensation, i-cyclization, i-aminolysis kanye ne-acylation, i-rivaroxaban engahluziwe iyatholakala, futhi i-rivaroxaban eqediwe iyacwengwa.
Ukulungiselela: Lo mkhiqizo uyithebhulethi ebomvu ehlanganiswe nefilimu.

Izinsiza:
Umgogodla wethebhulethi: i-microcrystalline cellulose, i-croscarmellose sodium, i-lactose monohydrate, i-hypromellose, i-sodium lauryl sulfate, i-magnesium stearate
Ukugqoka: i-polyethylene glycol, i-hypromellose, i-titanium dioxide, i-iron oxide ebomvu

I-Rivaroxaban iyisidakamizwa esikhethwa kakhulu, esithathwa ngomlomo esivimbela ngokuqondile i-factor Xa.Ngokuvinjelwa okukhetha kakhulu nokuncintisana kwe-factor Xa yamahhala nebophekile kanye nomsebenzi we-prothrombin, andisa ipuleti lesikhathi le-thromboplastin elicushiwe (PT) kanye nesikhathi se-prothrombin (aPTT) ngendlela encike kumthamo, engaphazamisa impophoma yokuhlangana. kuvimbela ukukhiqizwa kwe-thrombin ne-thrombosis.I-Rivaroxaban ayivimbeli i-thrombin (isici esisebenzayo Ⅱ), futhi ayizange ifakazele ukuthi inomthelela kumaplatelet.
Umehluko obalulekile phakathi kwe-rivaroxaban ne-fondaparinux/heparin ukuthi ayidingi ukubamba iqhaza kwe-antithrombin III futhi ingaphikisa ngokuqondile i-factor Xa yamahhala neboshiwe;kuyilapho i-heparin idinga i-antithrombin III ukuze isebenze, futhi Ayinawo umphumela ku-factor Xa ku-prothrombin complex.

Imikhiqizo yethu ibhekwa kabanzi futhi ithembekile kubasebenzisi bokugcina futhi ingahlangabezana nezidingo ezihlala zishintsha zezimali nezenhlalo ze-OEM Customized Rivaroxaban CAS No. ukuthambekela kokuthuthukiswa kwale mboni futhi ugcwalise injabulo yakho ngempumelelo.Kunoma ubani othathekayo ngaphakathi kwezixazululo zethu, kufanele uxhumane nathi ngokukhululekile.
I-OEM eyenziwe ngokwezifisoI-China Chemical and Pharmaceutical Raw Material, Sinezixazululo ezingcono kakhulu kanye nokuthengisa okufanelekayo kanye nethimba lobuchwepheshe.Ngokuthuthukiswa kwenkampani yethu, siyakwazi ukuletha amakhasimende imikhiqizo engcono kakhulu, ukusekelwa okuhle kwezobuchwepheshe, isevisi ephelele emva kokuthengisa.


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